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Table 1 Classification of epigenetic modifiers

From: Epigenetic regulation in cancer progression

Class

Enzymes

Histone Acetyltransferases (HATs)

ELP3/KAT9

PCAF/KAT2B

MORF/MYST4/KAT6B

GTF3C4

CBP/KAT3A

HBO1/MYST2/KAT7

HAT3

p300/KAT3B

MOF/MYST1/KAT8

HAT1/KAT1

Tip60/KAT5

KAT10

GCN5/KAT2A

MOZ/MYST3/KAT6A

TFIIIC90/KAT12

Histone Deacetylases (HDACs)

HDAC1

HDAC7

SIRT2

HDAC2

HDAC8

SIRT3

HDAC3

HDAC9

SIRT4

HDAC4

HDAC10

SIRT5

HDAC5

HDAC11

SIRT6

HDAC6

SIRT1

SIRT7

Histone Methyltransferases (HMTs)

ASH1

NSD1/KMT3B

SETD1A

Clr4/KMT1

PRMT1

SETD8/Pr-SET7/KMT5A

Dot1L/KMT4

PRMT3

SETDB1

EZH2/KMT6

PRMT4/CARM1

SETDB2/KMT1F/CLL8

G9a/EHMT2

PRMT5/JBP1

SMYD2/KMT3C

GLP/EHMT1

PRMT6

SUV39H1

KMT5B/KMT5C

Riz1/Riz2/KMT8

SUV39H2

MLL1

NF20

SUV4-20H2/KMT5C

MLL2

RNF40

TRX/ KMT2a

MLL3

SET1A

HIF-1/ SET2/HYPB/KMT3A

MLL4

SET1B

 

MLL5

SET7/9

 

Histone Demethylases (HDMs)

ARID1A

JHDM1b/FBXL10/KDM2B

JMJD2D/KDM4D

ARID5B

JHDM2A/KDM3A

JMJD3/KDM6B

JARID1A/RBBP2/KDM5A

JHDM3A/JMJD2A/KDM4A

LSD1/KDM1

JARID1B/PLU1/KDM5B

JMJD1A

LSD2

JARID1C/SMCX/KDM5C

JMJD1B/KDM3B

PHF2

JARID1D/SMCY/KDM5D

JMJD2A

PLU1

JHD1/KDM2

JMJD2B/KDM4B

UTX/KDM6A

JHDM1a/FBXL11/KDM2A

JMJD2C/GASC1/KDM4C

 

DNA Methyltransferases (DNMTs)

DNMT1

DNMT3b

DNMT1o

DNMT3a

DNMT3L

 

DNA Demethylases

TET1

TET2

TET3